Thursday 17 July 2025

Cetrorelix acetate is a synthetic decapeptide that is mainly used in assisted reproductive technology to prevent early ovulation in patients with controlled ovarian stimulation.Cetrorelix acetate, also commonly known as cetrorelix, is a gonadotropin-releasing hormone (GnRH) antagonist...

Thursday 17 July 2025

Ganirelix is a synthetic decapeptide compound whose acetate, Ganirelix Acetate, is a gonadotropin-releasing hormone (GnRH) receptor antagonist. The amino acid sequence is Ac-D-2Nal-D-4Cpa-D-3Pal-Ser-Tyr-D-HomoAr g(9,10-Et2)-Leu-L-HomoArg(9,10-Et2)-Pro- D-Ala-NH2.It is used clinically...

Thursday 17 July 2025

Degarelix acetate is a synthetic gonadotropin-releasing hormone (GnRH) receptor antagonist that exerts its anti-prostate cancer effects by reversibly binding to GnRH receptors in the pituitary gland, reducing the release of gonadotropins and testosterone. Brand: Soarwin EC Number...

Thursday 17 July 2025

Terlipressin is a new type of synthetic long-acting vasopressin preparation, belonging to a precursor drug, itself inactive, in vivo by the action of aminopeptidase, to remove its N-terminal 3 glycyl residues, slowly “release” the active lysine pressin. It is this “slow release”...

Thursday 17 July 2025

Cagrilintide is a novel long-acting acylated glucagon analogue under investigation as a non-selective agonist of the amygdalin receptor (AMYR) and calcitonin G-protein-coupled receptor (CChemicalbookTR).Cagrilintide significantly reduces body weight and decreases food intake.Cagrilintide...

Thursday 17 July 2025

Goserelin 是一种具有类似作用的促那瑞林类似物，于 1987 年在法国获准上市。戈舍瑞林是黄体生成素释放激素的类似物，长期使用本品可抑制垂体黄 体生成素的合成，从而引起男性血清睾酮和女性血清雌二醇的下降，停用此作用后可逆转， 初次使用本品可暂时增加男性血清睾酮浓度和女性血清雌二醇浓度。在男性患者中，血清睾 酮浓度在首次注射该药物后约 21 天降至贮库水平，并在随后的治疗中维持在这些水平，这导致大多数患者的前列腺肿瘤消退 和症状改善。在女性患者中，血清雌二醇浓度在初始给药后约 21 天受到抑制，并在后续治疗中每 28 天维持在绝经后水平。本品的半衰期为...